PerkinElmer

Receptor Ligand Binding

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Simplify the development of your assays and the calculation of your results using our radioligands, receptor-transfected cell membranes, and cell lines for radioligand binding applications.

Because radioligands can be directly detected, there is no need to generate intermediate antibodies against your target. Eliminating these antibodies also eliminates the need to optimize an antibody titer and reduces your total assay time by skipping intermediate incubation steps.

You’ll find our receptor-ligand binding reagents and related products perfect matches for all of your receptor binding studies.

 

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"Receptor Ligand Binding" 1-50 of 749 Products and Services

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MICROBETA FILTERMAT-24 CELL HARVESTER

Speed and simplicity are the primary strengths of the FilterMate Harvester. From beginning to end, the FilterMate system is easy to use. Need additional information? Click on the tabs in the product details section below.

UNIFILTER-24 CELL HARVESTER

Speed and simplicity are the primary strengths of the Unifilter Harvester.

UNIFILTER-96 CELL HARVESTER

Speed and simplicity are the primary strengths of the Unifilter Harvester.

UNIFILTER-96 CELL HARVESTER SS

Speed and simplicity are the primary strengths of the Unifilter Harvester.

MICROBETA FILTERMAT-96 CELL HARVESTER

Speed and simplicity are the primary strengths of the FilterMate Harvester. From beginning to end, the FilterMate system is easy to use.

OMNIFILTER-96 CELL HARVESTER

Speed and simplicity are the primary strengths of the OmniFilter Harvester.
LabChip EZ Reader

EZ READER, SHIP LEVEL

The EZ Reader can help to save time and money in your laboratory by identifying the most promising lead candidates faster.

The EZ Reader instrument is available outside the EU. Please contact your local representative for further information.

Cytisine HCl, [3,5-3H(N)]-, 25µCi (925kBq)

Cytisine HCl, [3,5-3H(N)]- will now be made available on a fresh lot schedule. NET1054025UC and NET1054250UC will be available as a fresh lot once a year on March 6 in 2017.
List Price : 690.00 CAD

Oxotremorine-M Acetate, [Methyl-3H]-,>97%, 250µCi (9.25MBq)

250 µCi quantities of tritiated oxotremorine-M are available for your research.
List Price : 2650.00 CAD
PerkinElmer

Membrane Target Systems: Cannabinoid CB1 (human) membrane preparation, in CHO-K1 cells. 400 Units.

Our Membrane Target System membranes are prepared from cells that express recombinant or endogenous receptors. Selected for optimal performance in binding assays.
List Price : 1100.00 CAD

Interleukin-1β (human, recombinant), [125I], 5µCi

NEX232 Interleukin-1 (IL-1) refers to a group of three polypeptides (interleukin-1 alpha (IL-1α), interleukin-1 beta (IL-1β) and interleukin-1 receptor antagonist (IL-1Ra)), that play a central role in the regulation of immune and inflammatory responses.

IL-1β is a pro-inflammatory cytokine involved in immune defense against infection.

List Price : 1150.00 CAD
PerkinElmer

Membrane Target Systems: Prokineticin PKR2 (human) membrane preparation

Cell membranes prepared from cells stably-transfected with human Prokineticin PKR2 receptor, in HEK-293 cells.
List Price : 1100.00 CAD
PerkinElmer

Anti-rabbit YSI 500 MG

Anti-rabbit-coated SPA beads, for capturing rabbit IgG antibodies in proximity-based radiometric scintillation assays.
List Price : 1150.00 CAD

Norepinephrine, Levo-[7-3H]-, 250µCi (9.25MBq)

250 µCi quantities of Levo-[7-3H]-Norepinephrine are available for your research. This product has a scheduled release date for the third Monday in July.
List Price : 1400.00 CAD

(-)-CGP-12177, [5,7-3H]-, 25µCi (925kBq)

25 µCi quantities of (-)-CGP-12177, [5,7-3H]- are available for your research.
List Price : 590.00 CAD

Cyclopentyl-1,3-Dipropylxanthine, 8-[Dipropyl-2,3-3H(N)]-, 250µCi (9.25MBq)

250 µCi quantities of Cyclopentyl-1, 3-Dipropylxanthine, 8-[Dipropyl-2, 3-3H(N)]- (DPCPX) are available for your research.
List Price : 1500.00 CAD
PerkinElmer

Glutathione YSI 50MG

Glutathione-coated SPA beads, for capturing GST-tagged proteins in proximity-based radiometric scintillation assays.
List Price : 1150.00 CAD
Receptor-expressing cell lines

ValiScreen Orexin 2 (OX2)-like (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.

QRFP-43, [125I], Human Radioligand, 10µCi (370kBq)

QRFP-43 is a 43 amino acid polypeptide starting from N-terminal pyroglutamic acid and ending at C-terminal arginine-phenylalanine-amide. The intravenous administration of QRFP-43 caused the release of aldosterone, suggesting that QRFP and its receptor have a regulatory function in the rat adrenal gland.
List Price : 1400.00 CAD
PerkinElmer

Streptavidin PVT 25 X 2G

Streptavidin-coated SPA beads, for capturing biotinylated biomolecules in proximity-based radiometric scintillation assays.
List Price : 75100.00 CAD

Interleukin-1β (human, recombinant), [125I], 10µCi

NEX232 Interleukin-1 (IL-1) refers to a group of three polypeptides (interleukin-1 alpha (IL-1α), interleukin-1 beta (IL-1β) and interleukin-1 receptor antagonist (IL-1Ra)), that play a central role in the regulation of immune and inflammatory responses.

IL-1β is a pro-inflammatory cytokine involved in immune defense against infection.

List Price : 2000.00 CAD

Sauvagine, [125I]-Tyr0], 10µCi

NEX306 [125I]Tyr0-Sauvagine has been shown to be active in receptor binding assays and has been used for receptor autoradiography.
List Price : 1200.00 CAD

Adenosine 3',5'-cyclic Phosphoric Acid, 2`-O-succinyl [125I]-Iodotyrosine Methyl Ester-, 1µCi

Adenosine 3',5'-cyclic Phosphoric Acid, 2'-O-succinyl, [125I]-Iodotyrosine Methyl Ester- Adenosine is an inhibitory neurotransmitter, believed to play a role in promoting sleep and suppressing arousal, with levels increasing with each hour an organism is awake.
List Price : 440.00 CAD
Receptor-expressing cell lines

ValiScreen Muscarinic M2 (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.
Receptor-expressing cell lines

ValiScreen Galanin Gal1 (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.

DAMGO, [Tyrosyl-3,5-3H(N)]-, 1mCi (37MBq)

1 mCi quantities of [Tyrosyl-3, 5-3H(N)]-DAMGO are available for your research.
List Price : 4950.00 CAD
List Price : 1100.00 CAD

Kainic acid, [Isopropenyl-3H]-, 25µCi (925kBq)

25 µCi quantities of tritiated Kainic acid are available for your research.
List Price : 660.00 CAD

Caffeine, [1-Methyl-14C]-, 50µCi (1.85MBq)

50 quantities of [1-Methyl-14C]-Caffeine are available for your research.
List Price : 950.00 CAD
PerkinElmer

Membrane Target Systems: Epidermal Growth Factor Receptor EGF membrane preparation

Cell membranes prepared from A431 cells containing human endogenous EGF receptor.
List Price : 1100.00 CAD
PerkinElmer

Membrane Target Systems: Adrenergic alpha 2A (human) membrane preparation, in CHO-K1 cells. 400 Units.

Our Membrane Target System membranes are prepared from cells that express recombinant or endogenous receptors. Selected for optimal performance in binding assays.
List Price : 1100.00 CAD

MDL105,519, [3H]

250 µCi quantities of [3H]-MDL105,519 are available for your research.
List Price : 3050.00 CAD

Ro 15-1788, [N-Methyl-3H]-, 1MC

1 mCi quantities of [N-Methyl-3H]-Ro 15-1788 are available for your research.
List Price : 5600.00 CAD

Thyroxine, ([125I]-T4), L-[125I]-, 250µCi (9.25MBq), Specific Activity: 135-165µCi (5.00-6.11MBq)/µg

NEX111 L-3,5-Diiodothyronine is radioiodinated with no carrier added 125I using a modification of the Hunter and Greenwood method and is purified by reversed phase HPLC.
List Price : 1150.00 CAD

ACTH (1-39) 23Tyr [125I], 50 µCi

[125I]ACTH is lyophilized from an acetic acid solution (0.1%) containing bovine serum albumin (0.25%), lactose (5%), L-cysteine hydrochloride (0.1%) and aprotinin (0.3TIU/ml).
List Price : 5500.00 CAD
List Price : 1150.00 CAD

PDGF [125I] (human) 25 µCi

NEX433 [125I]-PDGF BB homodimer has been shown to work in RIA and receptor studies, using CHO cell line transfected with human PDGF B receptor, and human artery smooth muscle cells.
List Price : 2400.00 CAD

QRFP-43, [125I], Human Radioligand, 25µCi (925kBq)

QRFP-43 is a 43 amino acid polypeptide starting from N-terminal pyroglutamic acid and ending at C-terminal arginine-phenylalanine-amide. The intravenous administration of QRFP-43 caused the release of aldosterone, suggesting that QRFP and its receptor have a regulatory function in the rat adrenal gland.
List Price : 3000.00 CAD
PerkinElmer

Streptavidin PVT 2G

Streptavidin-coated SPA beads, for capturing biotinylated biomolecules in proximity-based radiometric scintillation assays.
List Price : 14700.00 CAD

Oxytocin, [Tyrosyl-3,5-3H]-, 50µCi (1.85MBq)

50 µCi quantities of [Tyrosyl-3,5-3H]-Oxytocin are available for your research.
List Price : 1200.00 CAD

MK-801, (+)-[3-3H]-, 250µCi (9.25MBq)

250 µCi quantities of (+)-[3-3H]-MK-801 are available for your research.
List Price : 2500.00 CAD
PerkinElmer

WGA PVT SPA 2G

WGA-coated SPA beads, for capturing cell membranes in proximity-based radiometric scintillation assays.
List Price : 4500.00 CAD
PerkinElmer

Glutathione YSI 500MG SILICAT

Glutathione-coated SPA beads, for capturing GST-tagged proteins in proximity-based radiometric scintillation assays.
List Price : 11200.00 CAD

Angiotensin II, [125I]-Sar1, Ile8], 50µCi

NEX248 [125I]-Sar1-Ile8-Angiotensin II is an angiotensin receptor antagonist which binds to a single class of receptors. [125I]-Sar1-Ile8-Angiotensin II is useful for studying AII receptors when an antagonist ligand is preferred, for receptor localization studies using autoradiographic techniques and for drug screening programs.
List Price : 2650.00 CAD
PerkinElmer

Membrane Target Systems: Glutamate mGlu5a (human) membrane preparation, in CHO-K1 cells. 400 Units.

Our Membrane Target System membranes are prepared from cells that express recombinant or endogenous receptors. Selected for optimal performance in binding assays.
List Price : 1100.00 CAD

Citalopram, [N-Methyl-3H]-, 50µCi (1.85MBq)

50 µCi quantities of [N-Methyl-3H]-Citalopram are available for your research.
List Price : 1300.00 CAD
PerkinElmer

ProfilerPro Kinase Peptide Substrate 14, for LabChip EZ Reader

Fluorescently-labelled peptide substrate 14 for kinase assays (inhibiton, target discovery, lead optimization)
List Price : 720.00 CAD
PerkinElmer

Membrane Target Systems: Galanin Gal1 (human) membrane preparation, in CHO-K1 cells. 400 Units.

Our Membrane Target System membranes are prepared from cells that express recombinant or endogenous receptors. Selected for optimal performance in binding assays.
List Price : 1100.00 CAD
PerkinElmer

Membrane Target Systems: Serotonin 5HT-5A (human) membrane preparation, in CHO-K1 cells. 400 Units.

Our Membrane Target System membranes are prepared from cells that express recombinant or endogenous receptors. Selected for optimal performance in binding assays.
List Price : 1100.00 CAD

"Receptor Ligand Binding" 1-50 of 749 Products and Services

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