PerkinElmer

Receptor Ligand Binding

OF

Simplify the development of your assays and the calculation of your results using our radioligands, receptor-transfected cell membranes, and cell lines for radioligand binding applications.

Because radioligands can be directly detected, there is no need to generate intermediate antibodies against your target. Eliminating these antibodies also eliminates the need to optimize an antibody titer and reduces your total assay time by skipping intermediate incubation steps.

You’ll find our receptor-ligand binding reagents and related products perfect matches for all of your receptor binding studies.

 

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"Receptor Ligand Binding" 1-50 of 764 Products and Services

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MICROBETA FILTERMAT-96 CELL HARVESTER

Speed and simplicity are the primary strengths of the FilterMate Harvester. From beginning to end, the FilterMate system is easy to use.

UNIFILTER-24 CELL HARVESTER

Speed and simplicity are the primary strengths of the Unifilter Harvester.

OMNIFILTER-96 CELL HARVESTER

Speed and simplicity are the primary strengths of the OmniFilter Harvester.
LabChip EZ Reader

EZ READER, SHIP LEVEL

The EZ Reader can help to save time and money in your laboratory by identifying the most promising lead candidates faster.

MICROBETA FILTERMAT-24 CELL HARVESTER

Speed and simplicity are the primary strengths of the FilterMate Harvester. From beginning to end, the FilterMate system is easy to use. Need additional information? Click on the tabs in the product details section below.

UNIFILTER-96 CELL HARVESTER

Speed and simplicity are the primary strengths of the Unifilter Harvester.

UNIFILTER-96 CELL HARVESTER SS

Speed and simplicity are the primary strengths of the Unifilter Harvester.

(+/-)Epibatidine, [5,6-Bicycloheptyl-3H]-, 250µCi (9.25MBq)

250 µCi quantities of [+/-] [5, 6-Bicycloheptyl-3H]-Epibatidine are available for your research. 
List Price : 4700.00 CAD

Lysergic Acid Diethylamide, 2-[125I]iodo-(+), 10µCi

NEX199 Preparations have been shown to be active in binding to the serotonin receptors. LSD affects a large number of the G protein coupled receptors, including all dopamine receptor subtypes, and all adrenoreceptor subtypes, as well as many others. LSD binds to most serotonin receptor subtypes except for 5-HT3 and 5-HT4.
List Price : 1000.00 CAD

Lysergic Acid Diethylamide, 2-[125I]iodo-(+), 50µCi

NEX199 Preparations have been shown to be active in binding to the serotonin receptors. LSD affects a large number of the G protein coupled receptors, including all dopamine receptor subtypes, and all adrenoreceptor subtypes, as well as many others. LSD binds to most serotonin receptor subtypes except for 5-HT3 and 5-HT4.
List Price : 2450.00 CAD
List Price : 1250.00 CAD
PerkinElmer

Membrane Target Systems: Neuromedin U NMU2 (human) membrane preparation

Cell membranes prepared from cells stably-transfected with human Neuromedin U NMU2 receptor, in HEK-293 cells.
List Price : 1100.00 CAD

CCK-8(SULPHATED), [3H]PROPIONY, 50 µCi

50 µCi quantities of [3H]PROPIONY CCK-8(SULPHATED) are available for your research.
List Price : 1700.00 CAD
List Price : 3100.00 CAD
List Price : 1200.00 CAD
PerkinElmer

DELFIA® L*R binding buffer concentrate (10x), 250 mL

Buffer for DELFIA® time-resolved fluorescence (TRF) ligand binding assays.
List Price : 650.00 CAD
PerkinElmer

Membrane Target Systems: Relaxin RXFP4 (GPCR142) (human) membrane preparation, in CHO-K1 cells. 400 Units.

Our Membrane Target System membranes are prepared from cells that express recombinant or endogenous receptors. Selected for optimal performance in binding assays.
List Price : 1000.00 CAD

Kainic acid, [Isopropenyl-3H]-, 1 mCi (37MBq)

1 mCi quantities of tritiated Kainic acid are available for your research.
List Price : 6100.00 CAD
Receptor-expressing cell lines

ValiScreen Prolactin Rel. Peptide PRRP (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.
Receptor-expressing cell lines

ValiScreen Muscarinic M1 (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.

Somatostatin-14 (human, recombinant), Receptor Grade, 10 µCi

NEX446 Tyr11 Somatostatin-14 is radioiodinated with no-carrier-added 125I using amodified lactoperoxidase procedure and is purified by reversed phase HPLC. This method predominantly labels tyrosine residues.
List Price : 1050.00 CAD

Dihydroxyphenylethylamine [2,5,6,7,8-3H] (Dopamine)

Dopamine receptors have key roles in many processes, including the control of motivation, learning, and fine motor movement, as well as modulation of neuroendocrine signaling.
List Price : 2000.00 CAD

Astemizole, [O-Methyl-3H]-, 250µCi (9.25MBq)

Astemizole, [O-Methyl-3H]- will now be made available on a fresh lot schedule. NET1140025UC, NET1140250UC, and NET1140001MC will be available as a fresh lot twice a year on March 6 and August 7 in 2017.
List Price : 3600.00 CAD

Escitalopram, [N-methyl-3H]-

250 µCi quantities of tritiated Escitalopram are available for your research.
List Price : 4950.00 CAD

AB-MECA, [125I]-(4-Amino-3-[125I]iodobenzyl-5`-N-)-, 50µCi

AB-MECA is radioiodinated with no carrier added 125I using a modification of the Hunter and Greenwood method and is purified by reversed phase HPLC.
List Price : 2700.00 CAD

Apamin [125I]His18-NH2, 25µCi

NEX242 [125I]-Apamin is a K+ channel antagonist and can be used in the detection and quantification of K+ channel receptors. [125I]-Apamin has been used in receptor binding assays and in autoradiography.
List Price : 1050.00 CAD

WIN 35428, [N-Methyl-3H]-, 25µCi (925kBq)

25 µCi quantities of tritiated WIN 35428 are available for your research.
List Price : 820.00 CAD
Receptor-expressing cell lines

ValiScreen Prostanoid CRTH2 (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.
PerkinElmer

Anti-sheep YSI 500 MG

Anti-sheep-coated SPA beads, for capturing sheep IgG antibodies in proximity-based radiometric scintillation assays.
List Price : 1150.00 CAD
PerkinElmer

Membrane Target Systems: Neuropeptide NPFF1 (human) membrane preparation

Cell membranes prepared from cells stably-transfected with human Neuropeptide NPFF1 receptor, in CHO-K1 cells.
List Price : 1100.00 CAD

Vasopressin (8-L-Arginine), [Phenylalanyl-3,4,5-3H(N)]

25 µCi quantities of [Phenylalanyl-3,4,5-3H(N)]-Vasopressin (8-L-arginine) are available for your research.
List Price : 730.00 CAD
Receptor-expressing cell lines

ValiScreen Muscarinic M2 (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.

DELFIA Eu-Labeling kit (Eu-N1-ITC chelate), 0.2mg

DELFIA® Europium labeling kit for labeling your own biomolecules for use in DELFIA time-resolved fluorescence assays. The ITC chelate reacts with free amine groups in the target biomolecule.
List Price : 640.00 CAD

Strychnine, [Benzene-Ring-3H]-, 250µCi (9.25MBq)

250 µCi quantities of tritiated Strychnine are available for your research.
List Price : 2300.00 CAD

MK-801, (+)-[3-3H]-%, 25µCi (925kBq)

25 µCi quantities of (+)-[3-3H]-MK-801 are available for your research.
List Price : 750.00 CAD

Substance P, [125I]Tyr8], 10µCi

Substance P, [125I]Tyr8] is radioiodinated with no carrier added 125I by a lactoperoxidase procedure and is purified by reversed phase HPLC.
List Price : 1350.00 CAD
PerkinElmer

STREP PVT SPECIAL 25 X 500 MG

Streptavidin-coated SPA beads, for capturing biotinylated biomolecules in proximity-based radiometric scintillation assays.
List Price : 91900.00 CAD

Oxytocin, [Tyrosyl-3,5-3H]-, 50µCi (1.85MBq)

50 µCi quantities of [Tyrosyl-3,5-3H]-Oxytocin are available for your research.
List Price : 1200.00 CAD

Cyclopentyl-1,3-Dipropylxanthine, 8-[Dipropyl-2,3-3H(N)]-, 1mCi (37MBq)

1 mCi quantities of Cyclopentyl-1, 3-Dipropylxanthine, 8-[Dipropyl-2, 3-3H(N)]- (DPCPX) are available for your research.
List Price : 3450.00 CAD

Epidermal Growth Factor (Murine), [125I]-,50µCi

Epidermal growth factor or EGF is a growth factor that plays an important role in the regulation of cell growth, proliferation, and differentiation by binding to its receptor EGFR.
List Price : 2350.00 CAD

Spiperone (Spiroperidol), [Benzene ring-3H]-, 1mCi (37MBq)

1 mCi quantities of [Benzene ring-3H]-Spiperone (Spiroperidol) are available for your research.
List Price : 4100.00 CAD

Rauwolscine, [Methyl-3H]-, 250µCi (9.25MBq)

250 µCi quantities of tritiated Rauwolscine are available for your research.
List Price : 2000.00 CAD
PerkinElmer

ProfilerPro Kinase Selectivity Assay Plate Kit 1, for LabChip EZ Reader

Kit consist of matched pairs of 384-well kinase-assay and substrate plates. Each assay plate contains 24 different predispensed frozen kinases. Substrate plates contain the appropriate fluorescent labeled peptides and ATP.
List Price : 1850.00 CAD
Receptor-expressing cell lines

ValiScreen TRH (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.
PerkinElmer

Protein A YSI 500 MG

Protein A-coated SPA beads, for capturing antibodies in proximity-based radiometric scintillation assays.
List Price : 1150.00 CAD

Neurokinin A, ([125I]-Substance K, 10µCi

NEX252 [125I]-NKA is a radioiodinated tachykinin which binds selectively to NK-2 receptors. Typical lots have been tested in a specific NK-2 radioreceptor assay. We do not recommend its use in a radioimmunoassay. The presence of a non-oxidized methionine typically leads to low antibody binding.
List Price : 950.00 CAD

Lysergic Acid Diethylamide, 2-[125I]iodo-(+), 250µCi

NEX199 Preparations have been shown to be active in binding to the serotonin receptors. LSD affects a large number of the G protein coupled receptors, including all dopamine receptor subtypes, and all adrenoreceptor subtypes, as well as many others. LSD binds to most serotonin receptor subtypes except for 5-HT3 and 5-HT4.
List Price : 5600.00 CAD
Receptor-expressing cell lines

ValiScreen Angiotensin AT1 (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.

"Receptor Ligand Binding" 1-50 of 764 Products and Services

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