PerkinElmer

Receptor Ligand Binding

OF

Simplify the development of your assays and the calculation of your results using our radioligands, receptor-transfected cell membranes, and cell lines for radioligand binding applications.

Because radioligands can be directly detected, there is no need to generate intermediate antibodies against your target. Eliminating these antibodies also eliminates the need to optimize an antibody titer and reduces your total assay time by skipping intermediate incubation steps.

You’ll find our receptor-ligand binding reagents and related products perfect matches for all of your receptor binding studies.

 

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"Receptor Ligand Binding" 1-50 of 749 Products and Services

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LabChip EZ Reader

EZ READER, SHIP LEVEL

The EZ Reader can help to save time and money in your laboratory by identifying the most promising lead candidates faster.

The EZ Reader instrument is available outside the EU. Please contact your local representative for further information.

UNIFILTER-24 CELL HARVESTER

Speed and simplicity are the primary strengths of the Unifilter Harvester.

UNIFILTER-96 CELL HARVESTER

Speed and simplicity are the primary strengths of the Unifilter Harvester.

OMNIFILTER-96 CELL HARVESTER

Speed and simplicity are the primary strengths of the OmniFilter Harvester.

UNIFILTER-96 CELL HARVESTER SS

Speed and simplicity are the primary strengths of the Unifilter Harvester.

MICROBETA FILTERMAT-96 CELL HARVESTER

Speed and simplicity are the primary strengths of the FilterMate Harvester. From beginning to end, the FilterMate system is easy to use.

MICROBETA FILTERMAT-24 CELL HARVESTER

Speed and simplicity are the primary strengths of the FilterMate Harvester. From beginning to end, the FilterMate system is easy to use. Need additional information? Click on the tabs in the product details section below.

Lysergic Acid Diethylamide, 2-[125I]iodo-(+), 50µCi

NEX199 Preparations have been shown to be active in binding to the serotonin receptors. LSD affects a large number of the G protein coupled receptors, including all dopamine receptor subtypes, and all adrenoreceptor subtypes, as well as many others. LSD binds to most serotonin receptor subtypes except for 5-HT3 and 5-HT4.
List Price : 2450.00 CAD

(+/-)Epibatidine, [5,6-Bicycloheptyl-3H]-, 25µCi (925kBq)

25 µCi quantities of [+/-] [5, 6-Bicycloheptyl-3H]-Epibatidine are available for your research.
List Price : 2000.00 CAD

Lysergic Acid Diethylamide, 2-[125I]iodo-(+), 250µCi

NEX199 Preparations have been shown to be active in binding to the serotonin receptors. LSD affects a large number of the G protein coupled receptors, including all dopamine receptor subtypes, and all adrenoreceptor subtypes, as well as many others. LSD binds to most serotonin receptor subtypes except for 5-HT3 and 5-HT4.
List Price : 5600.00 CAD
List Price : 1250.00 CAD
List Price : 2050.00 CAD
List Price : 1450.00 CAD

Dihydroxyphenylethylamine [2,5,6,7,8-3H] (Dopamine)

Dopamine receptors have key roles in many processes, including the control of motivation, learning, and fine motor movement, as well as modulation of neuroendocrine signaling.
List Price : 2000.00 CAD

Norepinephrine, Levo-[ring-2,5,6-3H]-, 250µCi (9.25MBq)

250 µCi quantities of Levo-[ring-2, 5, 6-3H]-Norepinephrine are available for your research.
List Price : 1500.00 CAD

IL-6 (human, recombinant), [125I], 25µCi

NEX269 Interleukin-6 (IL-6) is a protein that in humans is encoded by the IL6 gene. IL-6 is an interleukin that acts as both a pro-inflammatory and anti-inflammatory cytokine. It is secreted by T cells and macrophages to stimulate immune response to trauma, especially burns or other tissue damage leading to inflammation.
List Price : 4800.00 CAD
PerkinElmer

ProfilerPro Kinase Peptide Substrate 10, for LabChip EZ Reader

Fluorescently-labelled peptide substrate 10 for kinase assays (inhibiton, target discovery, lead optimization)
List Price : 720.00 CAD

Somatostatin-14 (human, recombinant), Receptor Grade, 10 µCi

NEX446 Tyr11 Somatostatin-14 is radioiodinated with no-carrier-added 125I using amodified lactoperoxidase procedure and is purified by reversed phase HPLC. This method predominantly labels tyrosine residues.
List Price : 1050.00 CAD
Receptor-expressing cell lines

ValiScreen Adrenergic alpha 2B (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.
PerkinElmer

Glutathione YSI 500MG SILICAT

Glutathione-coated SPA beads, for capturing GST-tagged proteins in proximity-based radiometric scintillation assays.
List Price : 11200.00 CAD

Lysergic Acid Diethylamide, 2-[125I]iodo-(+), 10µCi

NEX199 Preparations have been shown to be active in binding to the serotonin receptors. LSD affects a large number of the G protein coupled receptors, including all dopamine receptor subtypes, and all adrenoreceptor subtypes, as well as many others. LSD binds to most serotonin receptor subtypes except for 5-HT3 and 5-HT4.
List Price : 1000.00 CAD
Receptor-expressing cell lines

ValiScreen Neuropeptide Y Y2 (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.
Receptor-expressing cell lines

Neuropeptide FF NPFF1 ValiScreen Cell Line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.

RTI-55, [125I]-, 25µCi (925kBq)

NEX272 [125I]-RTI-55 is an excellent radioligand for the study of the dopamine transporter sites using either tissue homogenates or autoradiographic methods--especially in regions of low receptor density.
List Price : 1050.00 CAD

MK-912, [3H(G)]

This compound replaces NET1059. MK-912 is an alpha-2 adrenoceptor antagonist. This novel alpha-2 adrenoceptor antagonist radioligand [3H]-MK912 may be used in studies of the regulation of cardiovascular and CNS function.
List Price : 3050.00 CAD

GLP-1 (7-36), [125I]-, 10µCi (370kBq)

NEX308 Glucagon-like peptide-1 (GLP-1) is derived from the transcription product of the proglucagon gene. The major source of GLP-1 in the body is the intestinal L cell that secretes GLP-1 as a gut hormone. The biologically active forms of GLP-1 are: GLP-1-(7-37) and GLP-1-(7-36)NH2.
List Price : 1400.00 CAD
PerkinElmer

ProfilerPro Kinase Selectivity Assay Plate Kit 1, for LabChip EZ Reader

Kit consist of matched pairs of 384-well kinase-assay and substrate plates. Each assay plate contains 24 different predispensed frozen kinases. Substrate plates contain the appropriate fluorescent labeled peptides and ATP.
List Price : 1850.00 CAD

Norepinephrine Hydrochloride, DL-[7-3H(N)]-, 250µCi (9.25MBq)

250 µCi quantities of DL-[7-3H(N)]-Norepinephrine Hydrochloride are available for your research.
List Price : 950.00 CAD
PerkinElmer

DELFIA® L*R binding buffer concentrate (10x), 250 mL

Buffer for DELFIA® time-resolved fluorescence (TRF) ligand binding assays.
List Price : 650.00 CAD
Receptor-expressing cell lines

ValiScreen Leukotriene BLT1 (LTB4R1) (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.

DTG (1,3-Di-o-tolylguanidine, [p-ring-3H]-), [5-3H(N)]-, 250µCi (9.25MBq)

250 µCi quantities of [5-3H(N)]-DTG (1, 3-Di-o-tolylguanidine, [p-ring-3H]-) are available for your research.
List Price : 2500.00 CAD
PerkinElmer

Membrane Target Systems: Serotonin 5HT-2C (e) (human) membrane preparation, in CHO-K1 cells. 400 Units.

Our Membrane Target System membranes are prepared from cells that express recombinant or endogenous receptors. Selected for optimal performance in binding assays.
List Price : 1100.00 CAD
PerkinElmer

ProfilerPro Kinase Peptide Substrate 7, for LabChip EZ Reader

Fluorescently-labelled peptide substrate 7 for kinase assays (inhibiton, target discovery, lead optimization)
List Price : 720.00 CAD
PerkinElmer

ProfilerPro Kinase Peptide Substrate 16, for LabChip EZ Reader

Fluorescently-labelled peptide substrate 16 for kinase assays (inhibiton, target discovery, lead optimization)
List Price : 720.00 CAD
PerkinElmer

Membrane Target Systems: Vasopressin V1b (human) membrane preparation, in CHO-K1 cells. 400 Units.

Cell membranes prepared from CHO-K1 cells stably-transfected with human Vasopressin V1b receptor, 400 units.
List Price : 1100.00 CAD
PerkinElmer

Membrane Target Systems: Galanin Gal1 (human) membrane preparation, in CHO-K1 cells. 400 Units.

Our Membrane Target System membranes are prepared from cells that express recombinant or endogenous receptors. Selected for optimal performance in binding assays.
List Price : 1100.00 CAD
PerkinElmer

Anti-mouse YSI 500 MG

Anti-mouse-coated SPA beads, for capturing mouse IgG antibodies in proximity-based radiometric scintillation assays.
List Price : 1400.00 CAD

Nociceptin, [Leucyl-3,4,5-3H], 50µCi (1.85MBq)

50 µCi quantities of [Leucyl-3, 4, 5-3H]-Nociceptin are available for your research.
List Price : 3700.00 CAD

QRFP-43, [125I], Human Radioligand, 25µCi (925kBq)

QRFP-43 is a 43 amino acid polypeptide starting from N-terminal pyroglutamic acid and ending at C-terminal arginine-phenylalanine-amide. The intravenous administration of QRFP-43 caused the release of aldosterone, suggesting that QRFP and its receptor have a regulatory function in the rat adrenal gland.
List Price : 3000.00 CAD
PerkinElmer

Membrane Target Systems: Neuropeptide NPFF2 (human) membrane preparation

Cell membranes prepared from cells stably-transfected with human Neuropeptide NPFF2 receptor, in CHO-K1 cells.
List Price : 1050.00 CAD
Receptor-expressing cell lines

ValiScreen Adrenergic beta 3 (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.
Receptor-expressing cell lines

ValiScreen Vasopressin V2 (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.

Neurotensin, [3,11-Tyrosyl-3,5-3H(N)]-, 250µCi (9.25MBq)

250 µCi quantities of [3, 11-Tyrosyl-3, 5-3H(N)]-Neurotensin are available for your research.
List Price : 3300.00 CAD

PDGF [125I] (human) 25 µCi

NEX433 [125I]-PDGF BB homodimer has been shown to work in RIA and receptor studies, using CHO cell line transfected with human PDGF B receptor, and human artery smooth muscle cells.
List Price : 2400.00 CAD
PerkinElmer

Membrane Target Systems: Adrenergic B2 (human) membrane preparation

Cell membranes prepared from cells stably-transfected with Adrenergic B2 (human) receptor, in HEK-293 cells.
List Price : 1100.00 CAD

CP 55940, [Side Chain-2,3,4-3H(N)]-, 1mCi (37MBq)

1 mCi quantities of [Side Chain-2, 3, 4-3H(N)]-CP 55940 are available for your research.
List Price : 5700.00 CAD
PerkinElmer

Streptavidin PVT 50MG

Streptavidin-coated SPA beads, for capturing biotinylated biomolecules in proximity-based radiometric scintillation assays.
List Price : 380.00 CAD
Receptor-expressing cell lines

ValiScreen TRH (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.
PerkinElmer

ProfilerPro Kinase Peptide Substrate 29, for LabChip EZ Reader

Fluorescently-labelled peptide substrate 29 for kinase assays (inhibiton, target discovery, lead optimization)
List Price : 720.00 CAD

Dihydroxyphenylethylamine, 3,4-[7-3H]-, 250µCi (9.25MBq)

250 µCi quantities of 3, 4-[7-3H]-Dihydroxyphenylethylamine (Dopamine) are available for your research.
List Price : 750.00 CAD

"Receptor Ligand Binding" 1-50 of 749 Products and Services

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